A Dose-Range Study of Aleniglipron (GSBR-1290) in Participants Living With Obesity or Overweight With at Least One Weight-related Comorbidity

Purpose

Phase 2 clinical study will evaluate the safety, tolerability, pharmacokinetics (PK), and efficacy of various aleniglipron (GSBR-1290) dose regimens compared with placebo in participants living with obesity or overweight with ≥ 1 weight-related comorbidity, in addition to diet and exercise, over a 44-week period.

Conditions

  • Obesity
  • Overweight
  • Chronic Weight Management

Eligibility

Eligible Ages
Between 18 Years and 79 Years
Eligible Sex
All
Accepts Healthy Volunteers
No

Inclusion Criteria

  • Signed informed consent - BMI ≥30 kg/m2 or BMI ≥27.0 kg/m2 and previous/current diagnosis of ≥ 1 obesity related comorbidity

Exclusion Criteria

  • Previous documented diagnosis of diabetes mellitus - Self-reported change in body weight >5% within 3 months before Screening - Have a prior or planned surgical treatment for obesity (excluding liposuction or abdominoplasty, if performed >1 year prior to screening) - Use of medications intended to promote weight loss, within 6 months prior to Screening

Study Design

Phase
Phase 2
Study Type
Interventional
Allocation
Randomized
Intervention Model
Parallel Assignment
Primary Purpose
Treatment
Masking
Triple (Participant, Care Provider, Investigator)

Arm Groups

ArmDescriptionAssigned Intervention
Experimental
Sentinel
Participants will receive aleniglipron or placebo administered orally.
  • Drug: aleniglipron or placebo
    Drug: aleniglipron administered orally; Drug: placebo administered orally
Experimental
Cohort 1a
Participants will receive aleniglipron or placebo administered orally.
  • Drug: aleniglipron or placebo
    Drug: aleniglipron administered orally; Drug: placebo administered orally
Experimental
Cohort 1b
Participants will receive aleniglipron or placebo administered orally.
  • Drug: aleniglipron or placebo
    Drug: aleniglipron administered orally; Drug: placebo administered orally
Experimental
Cohort 1c
Participants will receive aleniglipron or placebo administered orally.
  • Drug: aleniglipron or placebo
    Drug: aleniglipron administered orally; Drug: placebo administered orally

Recruiting Locations

More Details

NCT ID
NCT06703021
Status
Active, not recruiting
Sponsor
Gasherbrum Bio, Inc., a wholly owned subsidiary of Structure Therapeutics